SCHEMBL9259602

SCHEMBL9259602

COC(=O)CCc1ccc(-c2nc(-c3ccc(C(C)(C)N)cc3)cn2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.40
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
FFAR1 O14842 2/20 0.37
SYK P43405 3/20 0.36
AVPR1B P47901 3/20 0.36
TP53 P04637 1/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
CDK1 P06493 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257933 0.91 HRH3 (0.39) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9251406 0.88 RXRA (0.44) FFAR1PPARGPPARDPPARA
SCHEMBL9251212 0.87 HRH3 (0.42) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9248511 0.87 HRH3 (0.42) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9250844 0.84 HRH3 (0.42) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9259034 0.83 NPC1 (0.42) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9259613 0.83 HRH3 (0.40) HRH3AVPR1B
SCHEMBL9257434 0.83 NPC1 (0.42) HRH3NPC1RAB9AHPGDTSHR
SCHEMBL9255567 0.83 HRH3 (0.40) HRH3NPC1RAB9ASYKAVPR1B
SCHEMBL9256832 0.83 ACVR1 (0.41) HRH3HPGDTSHRHSD17B10PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed