SCHEMBL9256020

SCHEMBL9256020

C/C=C/COc1ccc(C(=O)Oc2ccc(F)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.45
MAPT P10636 3/20 0.45
MAOB P27338 3/20 0.44
MEN1 O00255 1/20 0.44
ATM Q13315 1/20 0.43
NR4A2 P43354 1/20 0.42
PARP10 Q53GL7 1/20 0.41
PRSS1 P07477 1/20 0.41
ACR P10323 1/20 0.41
NPC1 O15118 2/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
TTR P02766 1/20 0.41
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21065718 0.87 KMT2A (0.54) KMT2AMAPTMEN1PRSS1ACR
SCHEMBL9256854 0.86 PRSS1 (0.48) KMT2AMAPTMAOBMEN1ATM
SCHEMBL9282589 0.82 ADRB2 (0.47) KMT2AMAPTMAOBMEN1ATM
SCHEMBL12869645 0.80 MAPT (0.64) KMT2AMAPTMEN1NPC1LMNA
SCHEMBL2838573 0.79 KMT2A (0.61) KMT2AMAPTMEN1ATMPARP10
SCHEMBL29009176 0.79 KMT2A (0.61) KMT2AMAPTMEN1ATMPARP10
SCHEMBL10332262 0.79 MAPT (0.47) KMT2AMAPTMAOBMEN1ATM
SCHEMBL2838297 0.79 KMT2A (0.49) KMT2AMAPTMEN1ATMNPC1
SCHEMBL2838301 0.79 KMT2A (0.49) KMT2AMAPTMEN1ATMNPC1
SCHEMBL11059608 0.78 LSS (0.51) KMT2AMAPTPARP10NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
US-5013477-A Alkenylbicyclohexane liquid crystals HOFFMANN-LA ROCHE INC. (US) 1991-05-07 US disclosed