SCHEMBL9256689

SCHEMBL9256689

CC(=O)c1ccc(O)cc1N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.46
ALDH1A1 P00352 5/20 0.46
HPGD P15428 3/20 0.46
CYP3A4 P08684 1/20 0.46
MAPK1 P28482 1/20 0.46
CA12 O43570 4/20 0.45
CA1 P00915 4/20 0.45
CA2 P00918 4/20 0.45
CA7 P43166 4/20 0.45
CA9 Q16790 4/20 0.45
CA14 Q9ULX7 4/20 0.45
CES2 O00748 1/20 0.45
TSHR P16473 1/20 0.43
KDM4E B2RXH2 4/20 0.43
GLA P06280 3/20 0.43
GAA P10253 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 1/20 0.43
S1PR4 O95977 1/20 0.43
MIF P14174 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9174091 0.98 HSD17B1 (0.44) HSD17B1ALDH1A1HPGDCYP3A4MAPK1
Acetic Acid SCHEMBL9056173 0.96 CA12 (0.45) HSD17B1ALDH1A1HPGDCYP3A4MAPK1
SCHEMBL11840032 0.83 ALDH1A1 (0.46) HSD17B1ALDH1A1HPGDCYP3A4MAPK1
SCHEMBL440293 0.80 ALDH1A1 (0.61) ALDH1A1HPGDCYP3A4CA12CA1
SCHEMBL164897 0.80 CA12 (0.46) ALDH1A1HPGDMAPK1CA12CA1
SCHEMBL3181880 0.80 ALDH1A1 (0.47) ALDH1A1HPGDCYP3A4MAPK1KDM4E
SCHEMBL16520525 0.79 ALDH1A1 (0.55) HSD17B1ALDH1A1HPGDCYP3A4MAPK1
SCHEMBL4385594 0.78 ALDH1A1 (0.50) ALDH1A1HPGDCYP3A4MAPK1CA1
SCHEMBL12045429 0.78 PRKCI (0.58) ALDH1A1HPGDMAPK1KDM4EGLA
SCHEMBL30310763 0.78 ALDH1A1 (0.50) ALDH1A1HPGDCYP3A4MAPK1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276191-A Reacting phenol with a nitrile in presence of Lewis acid catalyst in nitroalkane solvent to produce aminoalkyl para-hydroxyphenyl ketone FINE ORGANICS LIMITED (GB) 1994-01-04 US claimed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP claimed
WO-2017072662-A1 ANTIBODY CONJUGATES COMPRISING TOLL-LIKE RECEPTOR AGONIST NOVARTIS AG (CH) 2017-05-04 WO disclosed
WO-2016071856-A1 AMATOXIN DERIVATIVES AND CONJUGATES THEREOF AS INHIBITORS OF RNA POLYMERASE NOVARTIS AG (CH) 2016-05-12 WO disclosed
WO-2015189791-A1 AURISTATIN DERIVATIVES AND CONJUGATES THEREOF NOVARTIS AG (CH) 2015-12-17 WO disclosed
US-20140302553-A1 BIOSYNTHETICALLY GENERATED PYRROLINE-CARBOXY-LYSINE AND SITE SPECIFIC PROTEIN MODIFICATIONS VIA CHEMICAL DERIVATIZATION OF PYRROLINE-CARBOXY-LYSINE AND PYRROLYSINE RESIDUES IRM LLC (BM) 2014-10-09 US disclosed
CN-101855224-B Equilibrative nucleoside transporter ENT1 inhibitors JANSSEN PHARMACEUTICA NV 2012-11-28 CN disclosed
CN-101855224-A Equilibrative nucleoside transporter ENT 1 inhibitors JANSSEN PHARMACEUTICA NV 2010-10-06 CN disclosed
EP-0431871-B1 A process for the preparation of ketones FINE ORGANICS LTD (GB) 1995-06-07 EP disclosed
US-5276191-A Reacting phenol with a nitrile in presence of Lewis acid catalyst in nitroalkane solvent to produce aminoalkyl para-hydroxyphenyl ketone FINE ORGANICS LIMITED (GB) 1994-01-04 US disclosed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP disclosed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP disclosed
US-3987047-A ANORETICS BOEHRINGER INGELHEIM GMBH (DT) 1976-10-19 US disclosed