SCHEMBL9256791

SCHEMBL9256791

CCc1c(NC(C)C)cccc1C(=O)NC

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 4/20 0.44
PLK1 P53350 2/20 0.41
GAA P10253 2/20 0.40
POLB P06746 1/20 0.37
CLCN2 P51788 1/20 0.37
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
PTK2 Q05397 1/20 0.35
MTNR1A P48039 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21454987 0.80 GAA (0.52) CXCR2PLK1GAAPOLBADRA1D
SCHEMBL20972350 0.79 PLK1 (0.50) CXCR2PLK1GAACLCN2MTNR1A
SCHEMBL9256777 0.77 CLCN2 (0.44) CXCR2PLK1GAACLCN2KMT2A
SCHEMBL14688165 0.76 PLK1 (0.47) PLK1GAAPOLBHSD17B10
SCHEMBL24603694 0.74 GAA (0.62) PLK1GAAKMT2AMEN1
SCHEMBL16884622 0.74 KMT2A (0.47) PLK1GAAPOLBKMT2A
SCHEMBL28864326 0.73 PLK1 (0.45) PLK1GAAPOLBCLCN2KMT2A
SCHEMBL21590264 0.72 GAA (0.44) CXCR2PLK1GAAADRA1DADRA1A
SCHEMBL27573602 0.71 CHRNB2 (0.49) PLK1GAAKMT2AMEN1
SCHEMBL14648299 0.71 L3MBTL1 (0.42) PLK1GAAPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0672032-A1 NOVEL PHENYLETHYL AND PHENYLPROPYLAMINES Astra Aktiebolag (SE) 1995-09-20 EP disclosed