SCHEMBL9256929

SCHEMBL9256929

Cc1cccc2ncc(-c3nnnn3C(C)C)c(=O)n12

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 15/20 0.39
HTT P42858 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9263794 0.83 HTT (0.40) HTTCYP1A2POLBCYP2C19
SCHEMBL9263856 0.80 HTT (0.38) HTTCYP1A2POLBCYP2C19
SCHEMBL9262840 0.80 SMN1; SMN2 (0.43) MAP3K5HTTTDP1CYP1A2POLB
SCHEMBL9255169 0.78 CYP1A2 (0.43) HTTCYP1A2CYP2C19
SCHEMBL9213645 0.77 HTT (0.37) HTTCYP1A2POLBCYP2C19
SCHEMBL9259026 0.75 ADORA2A (0.38) HTTCYP1A2CYP2C19MAPT
SCHEMBL9256348 0.73 MAPK1 (0.46) HTTCYP1A2CYP2C19MAPT
SCHEMBL9273126 0.72 HTT (0.40) HTTCYP1A2POLBCYP2C19
SCHEMBL9261024 0.72 MAPT (0.39) MAP3K5TDP1CYP1A2POLBCYP2C19
SCHEMBL10518789 0.70 HTT (0.51) HTTCYP1A2POLBCYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475000-A Antiulcer agents CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1995-12-12 US disclosed
EP-0641340-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO- 1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1995-03-08 EP disclosed
WO-1993004065-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-03-04 WO disclosed