SCHEMBL9213645

SCHEMBL9213645

Cc1cccc2ncc(-c3nnn(C(C)C)n3)c(=O)n12

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
AAK1 Q2M2I8 4/20 0.33
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
POLB P06746 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
PIK3CD O00329 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208224 0.83 SMN1; SMN2 (0.39) HTTKDM4EALDH1A1HPGD
SCHEMBL9215987 0.79 NPC1 (0.40) HTTNPC1RAB9AAAK1KDM4E
SCHEMBL9217834 0.79 HTT (0.36) HTTNPC1RAB9AALDH1A1CYP1A2
SCHEMBL9256929 0.77 MAP3K5 (0.39) HTTCYP1A2POLBCYP2C19
SCHEMBL9259873 0.76 TRPV1 (0.38)
SCHEMBL9255180 0.72 MAPT (0.38) NPC1RAB9AAAK1KDM4EALDH1A1
SCHEMBL9263794 0.72 HTT (0.40) HTTKDM4EALDH1A1CYP1A2POLB
SCHEMBL9263856 0.69 HTT (0.38) HTTKDM4EALDH1A1CYP1A2POLB
SCHEMBL10518789 0.69 HTT (0.51) HTTNPC1RAB9AKDM4EALDH1A1
SCHEMBL9273126 0.68 HTT (0.40) HTTKDM4EALDH1A1CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475000-A Antiulcer agents CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1995-12-12 US disclosed
EP-0641340-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO- 1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1995-03-08 EP disclosed
WO-1993004065-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-03-04 WO disclosed