SCHEMBL9257052

SCHEMBL9257052

Cn1c(-c2ccc(C(C)(C)N)cc2)nc2cc(C(=O)NCCC(=O)O)ccc21

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.54
HDAC8 Q9BY41 3/20 0.54
HDAC6 Q9UBN7 3/20 0.54
HDAC3 O15379 2/20 0.50
HDAC2 Q92769 2/20 0.50
GCGR P47871 13/20 0.47
NAMPT P43490 1/20 0.46
JAK2 O60674 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
JAK3 P52333 1/20 0.46
PTGER4 P35408 1/20 0.44
PRSS12 P56730 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249604 0.90 HDAC1 (0.50) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9249490 0.86 HDAC1 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9247609 0.86 HDAC6 (0.56) HDAC1HDAC8HDAC6HDAC3HDAC2
Bromide SCHEMBL9253343 0.85 HDAC6 (0.55) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9255709 0.83 HDAC6 (0.55) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251361 0.83 HDAC6 (0.55) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9257057 0.83 HDAC6 (0.53) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9254127 0.83 HDAC6 (0.53) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9251340 0.82 HDAC1 (0.49) HDAC1HDAC8HDAC6HDAC3HDAC2
SCHEMBL9253539 0.81 HDAC1 (0.51) HDAC1HDAC8HDAC6HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed