SCHEMBL9257429

SCHEMBL9257429

N#Cc1ccc(Cc2cncs2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.49
LTA4H P09960 1/20 0.48
CYP11B1 P15538 9/20 0.43
CYP11B2 P19099 9/20 0.43
LOXL2 Q9Y4K0 2/20 0.43
CYP2A6 P11509 1/20 0.41
CYP19A1 P11511 4/20 0.40
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28752735 0.77 EPHX2 (0.50) HRH3LTA4HHPGD
SCHEMBL9710124 0.77 CYP3A4 (0.48) HRH3LTA4HCYP11B1CYP11B2LOXL2
SCHEMBL765420 0.77 SLC6A3 (0.51) LTA4HLOXL2KDM4EALDH1A1HPGD
SCHEMBL9389496 0.76 SLC6A3 (0.49) LTA4H
SCHEMBL24768074 0.72 SLC6A3 (0.55) LTA4HKDM4EALDH1A1CYP2D6HPGD
SCHEMBL1344068 0.72 LOXL2 (0.65) HRH3LOXL2CYP2A6CYP19A1SAE1
SCHEMBL28677901 0.71 LOXL2 (0.46) HRH3LTA4HLOXL2CYP2A6SAE1
SCHEMBL18892957 0.71 MYC (0.50) CYP11B2LOXL2CYP2A6CYP19A1ALDH1A1
SCHEMBL4009961 0.70 EPHX2 (0.64) HRH3CYP11B1CYP11B2LOXL2CYP2A6
SCHEMBL9267704 0.70 HRH3 (0.43) HRH3CYP11B1CYP11B2LOXL2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378721-A AROMATASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1995-01-03 US disclosed
US-5246952-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1993-09-21 US disclosed
EP-0477141-A1 Heteroarylmethylbenzols aromatase inhibitors CIBA-GEIGY AG (CH) 1992-03-25 EP disclosed