SCHEMBL9257792

SCHEMBL9257792

COC(=O)CCc1ccc(-c2nc(-c3ccc(C#N)cc3)c[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
MAPT P10636 4/20 0.40
POLB P06746 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
PTGES O14684 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
EP300 Q09472 4/20 0.37
HAT1 O14929 3/20 0.37
HRH3 Q9Y5N1 1/20 0.36
MMP12 P39900 1/20 0.36
MMP13 P45452 1/20 0.36
CXCR2 P25025 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3628694 0.82 CYP11B1 (0.56) CYP11B1CYP11B2MAPTPOLBEGLN1
SCHEMBL9568559 0.81 F2 (0.41) HDAC1
SCHEMBL9257084 0.81 F2 (0.41) HDAC1
Hydrochloric Acid SCHEMBL9254356 0.81 F2 (0.40) HDAC1
Hydrochloric Acid SCHEMBL3628690 0.80 CYP11B1 (0.55) CYP11B1CYP11B2MAPTPOLBEGLN1
SCHEMBL1338556 0.80 CYP11B1 (0.60) CYP11B1CYP11B2MAPTPOLBALDH1A1
SCHEMBL22756135 0.80 P2RY10 (0.45) LMNAHDAC6
SCHEMBL9259632 0.80 CYP11B1 (0.47) CYP11B1CYP11B2MAPTPOLBEGLN1
SCHEMBL8863941 0.80 CYP11B1 (0.42) CYP11B1CYP11B2MAPTPOLBEGLN1
SCHEMBL9259285 0.80 HRH3 (0.35) PTGESALDH1A1KDM4ELMNAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed