SCHEMBL9259632

SCHEMBL9259632

COC(=O)CCc1ccc(-c2nc(-c3ccc(C#N)cc3)n[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
S1PR1 P21453 1/20 0.42
VNN1 O95497 1/20 0.40
TRPA1 O75762 1/20 0.39
DGAT1 O75907 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
NR1H2 P55055 2/20 0.38
NR1H3 Q13133 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPK8 P45983 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
ABCB1 P08183 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254667 0.82 F2 (0.41) DGAT1ADORA3ADORA2ANR1H2NR1H3
SCHEMBL3628694 0.82 CYP11B1 (0.56) CYP11B1CYP11B2MAPTPOLBALDH1A1
Hydrochloric Acid SCHEMBL3628690 0.80 CYP11B1 (0.55) CYP11B1CYP11B2MAPTPOLBALDH1A1
SCHEMBL1338556 0.80 CYP11B1 (0.60) CYP11B1CYP11B2MAPTPOLBALDH1A1
SCHEMBL9257792 0.80 CYP11B1 (0.47) CYP11B1CYP11B2MAPTPOLBKDM4E
SCHEMBL9253364 0.77 CYP11B1 (0.52) CYP11B1CYP11B2MAPTPOLBKDM4E
SCHEMBL9250823 0.76 CDC25A (0.52) CYP11B1CYP11B2MAPTPOLBKDM4E
SCHEMBL9251931 0.76 CYP11B1 (0.52) CYP11B1CYP11B2MAPTPOLBKDM4E
SCHEMBL9251061 0.76 CYP11B1 (0.52) CYP11B1CYP11B2MAPTPOLBS1PR1
SCHEMBL9253975 0.74 HPGD (0.49) CYP11B1CYP11B2MAPTPOLBS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed