SCHEMBL9257868

SCHEMBL9257868

C#CC1Cc2ccccc2C1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
IDO1 P14902 2/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
PLAU P00749 1/20 0.38
DRD2 P14416 1/20 0.35
ANPEP P15144 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9123705 0.84 MAOA (0.50) MAOAMAOBPLAUANPEP
SCHEMBL29539739 0.74 IDO1 (0.41) IDO1PLAUANPEPDRD3
SCHEMBL385635 0.74 IDO1 (0.41) IDO1PLAUANPEP
SCHEMBL1415621 0.74 IDO1 (0.41) IDO1PLAUANPEPDRD3
SCHEMBL2725956 0.66 CYP1A2 (0.51) MAOAMAOBPLAUANPEP
SCHEMBL691835 0.66 PLAU (0.50) MAOAMAOBPLAUANPEP
SCHEMBL23978878 0.64 IDO1 (0.47) IDO1MAOAMAOBDRD2
SCHEMBL7332248 0.63 FAAH (0.47) IDO1ANPEP
SCHEMBL5870921 0.63 IDO1 (0.46) IDO1PLAUANPEPDRD3
SCHEMBL20095994 0.63 ANPEP (0.56) IDO1PLAUANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490772-B1 1,4-Disubstituted piperazines, their process of preparation and pharmaceutical compositions containing them ADIR (FR) 1995-07-26 EP disclosed