SCHEMBL9257875

SCHEMBL9257875

CCCCC1C/C(=C\c2ccccc2)C(=O)O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 6/20 0.47
CLK1 P49759 1/20 0.42
DYRK1A Q13627 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
CYP1A2 P05177 2/20 0.40
ALDH1A1 P00352 3/20 0.40
F3 P13726 1/20 0.38
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
AKT3 Q9Y243 1/20 0.38
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
MDM2 Q00987 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PPARG P37231 1/20 0.37
HTT P42858 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257881 1.00 GRM2 (0.47) GRM2CLK1DYRK1ADYRK1BCYP1A2
SCHEMBL7996076 0.85 DYRK1A (0.62) GRM2CLK1DYRK1ADYRK1BCYP1A2
SCHEMBL983907 0.85 CYP1A2 (0.49) CLK1DYRK1ADYRK1BCYP1A2ALDH1A1
SCHEMBL9252871 0.83 USP18 (0.48) CLK1DYRK1ADYRK1BALDH1A1MEN1
SCHEMBL9252868 0.83 USP18 (0.48) CLK1DYRK1ADYRK1BALDH1A1MEN1
SCHEMBL7992606 0.80 MAPT (0.50) CLK1DYRK1ADYRK1BCYP1A2ALDH1A1
SCHEMBL9253106 0.77 GRM2 (0.39) GRM2CYP1A2PPARGSIRT2
SCHEMBL9261410 0.76 PRKCA (0.43) GRM2CYP1A2PPARGSIRT2
SCHEMBL9261402 0.76 PRKCA (0.43) GRM2CYP1A2PPARGSIRT2
SCHEMBL981312 0.73 DYRK1A (0.69) CLK1DYRK1ADYRK1BCYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5416224-A Reaction of acetyldihydro-2-(3H)-furanone with aldehyde and alkali metal hydroxide HENKEL CORPORATION (US) 1995-05-16 US disclosed
EP-0559789-A1 PROCESS FOR THE PREPARATION OF $g(a)-ALKYL LACTONES HENKEL CORPORATION (US) 1993-09-15 EP disclosed
US-5231192-A Reacting an a-acyl lactone, an aldehyde and an alkali metal hydroxide; hydrogenation HENKEL CORPORATION (US) 1993-07-27 US disclosed
WO-1992010487-A1 PROCESS FOR CONVERTING α-ACYL-SUBSTITUTED LACTONES TO α-ALKYLIDENE-SUBSTITUTED LACTONES HENKEL CORPORATION (US) 1992-06-25 WO disclosed
WO-1992009590-A1 PROCESS FOR THE PREPARATION OF α-ALKYL LACTONES HENKEL CORPORATION (US) 1992-06-11 WO disclosed
US-4980342-A Process for the preparation of α-alkyl lactones HENKEL CORPORATION (US) 1990-12-25 US disclosed