SCHEMBL9258336

SCHEMBL9258336

CC(C)(C)OC(=O)N1CCC(C(=O)c2nc3ccccc3n2CCCCCC#N)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 1/20 0.42
NOD1 Q9Y239 1/20 0.42
STS P08842 2/20 0.42
HRH1 P35367 3/20 0.41
TACR2 P21452 1/20 0.41
TACR1 P25103 1/20 0.41
TP53 P04637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CNR2 P34972 3/20 0.40
CCR5 P51681 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OGFRL1 Q5TC84 1/20 0.40
GPR119 Q8TDV5 3/20 0.38
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
PTPN6 P29350 1/20 0.38
HIF1A Q16665 1/20 0.38
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9266382 0.99 NOD2 (0.43) NOD2NOD1STSHRH1TACR2
SCHEMBL13317058 0.84 KDM4E (0.54) NOD2NOD1STSHRH1TACR2
SCHEMBL9259877 0.83 HRH1 (0.49) HRH1TACR2TACR1TP53HSD17B10
SCHEMBL9260913 0.82 HRH1 (0.51) NOD2NOD1STSHRH1KDM4E
SCHEMBL9260703 0.81 HRH1 (0.42) HRH1TACR2TACR1TP53HSD17B10
SCHEMBL7899281 0.81 HRH1 (0.54) NOD2NOD1STSHRH1TACR2
SCHEMBL9268629 0.80 HRH1 (0.45) HRH1TACR2TACR1TP53HSD17B10
SCHEMBL7473405 0.80 HRH1 (0.44) NOD2NOD1STSHRH1TACR2
SCHEMBL9268701 0.80 HRH1 (0.53) HRH1TACR2TACR1
SCHEMBL9262955 0.80 HSD17B10 (0.44) HRH1TACR2TACR1TP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed