SCHEMBL9258632

SCHEMBL9258632

CN1CCC(C(O)c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 13/20 0.56
CYP2D6 P10635 12/20 0.56
KCNH2 Q12809 7/20 0.56
CHRM1 P11229 5/20 0.56
RAB9A P51151 1/20 0.53
ALOX5AP P20292 1/20 0.53
TP53 P04637 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695586 0.88 KCNH2 (0.51) HRH1CYP2D6KCNH2CHRM1RAB9A
Hydrochloric Acid SCHEMBL9543210 0.86 HRH1 (0.55) HRH1CYP2D6KCNH2CHRM1RAB9A
SCHEMBL9695626 0.86 KCNH2 (0.61) HRH1CYP2D6KCNH2CHRM1RAB9A
SCHEMBL9696761 0.85 CYP2D6 (0.43) HRH1CYP2D6KCNH2CHRM1RAB9A
SCHEMBL15569367 0.85 KCNH2 (0.51) HRH1CYP2D6KCNH2RAB9AALOX5AP
SCHEMBL9445676 0.84 HRH1 (0.68) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL9697130 0.82 KCNH2 (0.48) HRH1CYP2D6KCNH2CHRM1ALOX5AP
SCHEMBL9696461 0.81 GAA (0.49) HRH1CYP2D6KCNH2CHRM1TP53
SCHEMBL9445684 0.81 HRH1 (0.49) HRH1CYP2D6KCNH2CHRM1RAB9A
SCHEMBL9697133 0.80 ALDH1A1 (0.48) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed
WO-1992006086-A1 NOVEL 4-PIPERIDINYLCARBONYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1992-04-16 WO disclosed