SCHEMBL15569367

SCHEMBL15569367

O=C(c1ccccc1)N1CCC(C(O)c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.51
HRH3 Q9Y5N1 9/20 0.49
TP53 P04637 1/20 0.49
CYP2D6 P10635 2/20 0.47
HRH1 P35367 2/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SSTR5 P35346 1/20 0.46
ALOX5AP P20292 1/20 0.46
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9258632 0.85 HRH1 (0.56) KCNH2TP53CYP2D6HRH1RAB9A
SCHEMBL9695626 0.82 KCNH2 (0.61) KCNH2TP53CYP2D6HRH1RAB9A
SCHEMBL9695586 0.82 KCNH2 (0.51) KCNH2HRH3TP53CYP2D6HRH1
SCHEMBL15568226 0.82 HRH1 (0.63) KCNH2HRH3HRH1
SCHEMBL9696461 0.78 GAA (0.49) KCNH2HRH3TP53CYP2D6HRH1
SCHEMBL8227397 0.77 HRH1 (0.47) KCNH2TP53CYP2D6HRH1MEN1
SCHEMBL9445676 0.77 HRH1 (0.68) KCNH2HRH3TP53CYP2D6HRH1
SCHEMBL9697130 0.77 KCNH2 (0.48) KCNH2HRH3TP53CYP2D6HRH1
SCHEMBL9696448 0.76 P2RX7 (0.48) KCNH2HRH3TP53CYP2D6HRH1
SCHEMBL13108349 0.75 HSD11B1 (0.61) CYP2D6NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO claimed
WO-2014027053-A1 BENZIMIDAZOLES FOR THE TREATMENT OF CANCER MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2014-02-20 WO disclosed