SCHEMBL9258766

SCHEMBL9258766

COc1cccc2cc3n(c12)C(=O)CC3

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.51
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
CYP19A1 P11511 1/20 0.40
NQO2 P16083 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
KDM4E B2RXH2 4/20 0.38
HTT P42858 2/20 0.38
HCRTR2 O43614 5/20 0.38
HCRTR1 O43613 4/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MAPT P10636 2/20 0.37
CYP2A6 P11509 1/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018386 0.81 NOTUM (0.43) NOTUMHTR2AHTR2CCYP19A1NQO2
SCHEMBL9279199 0.80 NOTUM (0.56) NOTUMMEN1KMT2AALDH1A1MAPT
SCHEMBL9287309 0.73 NOTUM (0.51) NOTUMMEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL5774338 0.70 NOTUM (0.41) NOTUMSMN1; SMN2NPC1GAA
SCHEMBL9259627 0.68 NOTUM (1.00) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL30615209 0.68 NOTUM (1.00) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL9261564 0.68 NOTUM (0.57) NOTUMHTR2AHTR2CMEN1KMT2A
SCHEMBL9264812 0.68 NOTUM (0.57) NOTUMHTR2AHTR2CCYP19A1SMN1; SMN2
SCHEMBL26837191 0.68 HTR2A (0.59) HTR2AHTR2CDRD3KCNH2ALDH1A1
SCHEMBL13711870 0.66 HTR2A (0.60) HTR2AHTR2CCYP19A1NQO2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed
EP-0441517-A2 Tricyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1991-08-14 EP disclosed