SCHEMBL9258963

SCHEMBL9258963

COC(=O)COC(C)n1c(C(=O)C2CCN(CCCCC#N)CC2)nc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 7/20 0.42
TACR2 P21452 1/20 0.42
TACR1 P25103 1/20 0.42
KCNH2 Q12809 2/20 0.39
HTR4 Q13639 2/20 0.36
MCHR1 Q99705 7/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260700 0.85 HRH1 (0.42) HRH1TACR2TACR1ALDH1A1HPGD
SCHEMBL9268748 0.85 HRH1 (0.41) HRH1TACR2TACR1MCHR1ALDH1A1
SCHEMBL9261710 0.84 HRH1 (0.40) HRH1TACR2TACR1KCNH2HTR4
SCHEMBL9258610 0.81 KDM4E (0.39) HRH1TACR2TACR1HTR4MCHR1
SCHEMBL9259877 0.80 HRH1 (0.49) HRH1TACR2TACR1KCNH2MCHR1
SCHEMBL9259439 0.79 STS (0.44) ALDH1A1
SCHEMBL9258971 0.78 HRH1 (0.42) HRH1TACR2TACR1KCNH2MCHR1
SCHEMBL9267223 0.76 HRH1 (0.47) HRH1TACR2TACR1KCNH2MCHR1
SCHEMBL9268701 0.76 HRH1 (0.53) HRH1TACR2TACR1KCNH2
SCHEMBL9264785 0.76 HRH1 (0.39) HRH1TACR2TACR1KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed