SCHEMBL9259276

SCHEMBL9259276

CCC(Br)(C(=O)O)c1ccc(C#N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.44
EPHX2 P34913 1/20 0.43
KIF11 P52732 2/20 0.43
CTBP2 P56545 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP19A1 P11511 1/20 0.41
MLYCD O95822 1/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
HTT P42858 1/20 0.40
MAPT P10636 2/20 0.39
PTPN5 P54829 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MMP2 P08253 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7868519 0.82 EPHX2 (0.43) GSK3BEPHX2KIF11CTBP2CYP2A6
SCHEMBL7412854 0.79 MEN1 (0.63) GSK3BEPHX2KIF11CTBP2CYP2A6
SCHEMBL262672 0.77 CYP2C19 (0.47) KIF11HTTMAPTALDH1A1MEN1
SCHEMBL8224210 0.76 KIF11 (0.52) GSK3BEPHX2KIF11CYP2A6CA1
SCHEMBL10347288 0.76 MIF (0.50) GSK3BCYP19A1HTTMAPTALDH1A1
SCHEMBL6245761 0.74 KIF11 (0.50) EPHX2KIF11CYP2A6MLYCDCA1
SCHEMBL28846139 0.73 KIF11 (0.48) EPHX2KIF11CYP19A1MLYCDCA1
SCHEMBL12004125 0.72 KIF11 (0.52) KIF11CYP19A1MLYCDCA1CA2
SCHEMBL11622599 0.71 KIF11 (0.47) KIF11CYP2A6CYP19A1PTPN5MEN1
SCHEMBL31294502 0.71 KIF11 (0.47) GSK3BEPHX2KIF11CTBP2MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428160-A Condensation of imidazole derivative with cyano- or halo-substituted benzene derivative containing leaving group esterified with carboxylic or sulfonic acid CIBA-GEIGY CORPORATION (US) 1995-06-27 US disclosed
US-4889861-A Substituted imidazo[1,5-a]pyridine derivatives and other substituted bicyclic derivatives and their use as aromatase inhibitors CIBA-GEIGY CORP. (US) 1989-12-26 US disclosed
US-4728645-A THROMBOXANE SYNTHETASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1988-03-01 US disclosed