SCHEMBL9259487

SCHEMBL9259487

Clc1ccc(-c2nn(CCn3ccnc3)c3ccncc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.44
CYP19A1 P11511 2/20 0.43
CYP2A6 P11509 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
CYP2B6 P20813 1/20 0.43
AOC2 O75106 1/20 0.43
KCNH2 Q12809 1/20 0.43
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
QPCT Q16769 1/20 0.38
SCN1A P35498 1/20 0.38
SCN4A P35499 1/20 0.38
SCN5A Q14524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9255098 0.89 MAPK1 (0.41) KDM4EAOC2ALDH1A1SCN1ASCN4A
SCHEMBL9257071 0.88 CYP11B1 (0.47) KDM4ETSHRCYP19A1CYP11B1CYP11B2
SCHEMBL9302703 0.81 CSNK2A2 (0.39) KCNH2ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8135725 0.79 LTA4H (0.39) KDM4ETSHRKCNH2ALDH1A1CYP1A2
SCHEMBL9264220 0.78 KCNH2 (0.37) TP53KCNH2ALDH1A1MAPK1
SCHEMBL8138744 0.78 CYP2D6 (0.42) KCNH2ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9305127 0.78 MERTK (0.41) KDM4ETSHRKCNH2ALDH1A1CYP1A2
SCHEMBL8136501 0.78 MAPT (0.40) TP53
SCHEMBL8137068 0.76 CYP2D6 (0.49) KDM4ETSHRKCNH2CYP1A2CYP3A4
SCHEMBL8135688 0.76 MAPT (0.39) TP53KDM4ETSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed
US-5428169-A Antidepressants, treating compulsive disorders, stuttering, trichotillomania HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-06-27 US disclosed
US-5380847-A Reaction of 1-methylpiperidine-4-hydrazine, ketone and titanium isopropoxide to form hydrazone HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1995-01-10 US disclosed
EP-0594001-A1 Pyrazolo 4,3-c pyridines, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-27 EP disclosed
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US disclosed
US-5264576-A Antiserotonin agents, antidepressants and obsessive-compulsive disorders HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-11-23 US disclosed