SCHEMBL9259533

SCHEMBL9259533

O=c1[nH]c2ccccc2n2cc(-c3ccc(Cl)cc3)nc12

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.59
TAOK1 Q7L7X3 1/20 0.59
PBK Q96KB5 1/20 0.59
SLK Q9H2G2 1/20 0.59
ADORA2A P29274 1/20 0.51
ADORA3 P0DMS8 6/20 0.49
POLB P06746 2/20 0.48
KDM4E B2RXH2 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
PARP1 P09874 2/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9256388 0.89 ADORA3 (0.55) MAP4K4TAOK1PBKSLKADORA2A
SCHEMBL9255705 0.87 ADORA1 (0.51) MAP4K4TAOK1PBKSLKADORA2A
SCHEMBL9265209 0.87 POLB (0.48) MAP4K4TAOK1PBKSLKADORA3
SCHEMBL9264849 0.86 MAP4K4 (0.54) MAP4K4TAOK1PBKSLKADORA2A
SCHEMBL9256089 0.81 ADORA3 (0.54) MAP4K4ADORA2AADORA3POLBKDM4E
SCHEMBL9261950 0.79 ADORA3 (0.49) MAP4K4TAOK1PBKSLKADORA3
SCHEMBL9262896 0.79 ADORA3 (0.49) MAP4K4TAOK1PBKSLKADORA3
SCHEMBL9258369 0.76 POLB (0.48) ADORA3POLBPARP1GABRA1GABRA5
SCHEMBL9262609 0.76 DCLK1 (0.65) MAP4K4ADORA2AADORA3RAB9AGABRA1
SCHEMBL9538661 0.76 NPC1 (0.50) MAP4K4TAOK1PBKSLKADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993004066-A1 CERTAIN IMIDAZOQUINOXALINOLS; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-03-04 WO claimed
US-5182386-A G-Aminobutyric Acid NEUROGEN CORPORATION (US) 1993-01-26 US claimed
US-5473073-A Useful in diagnosis or treatment of anxiety, sleep and seizure disorders, overdose with bezodiazepine drug and memory enhancement NEUROGEN CORPORATION (US) 1995-12-05 US disclosed
WO-1993004066-A1 CERTAIN IMIDAZOQUINOXALINOLS; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-03-04 WO disclosed