SCHEMBL9255705

SCHEMBL9255705

Cc1ccc(-c2cn3c(n2)c(=O)[nH]c2ccccc23)cc1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.51
ADORA2A P29274 1/20 0.51
ADORA3 P0DMS8 6/20 0.49
POLB P06746 2/20 0.48
KDM4E B2RXH2 3/20 0.47
RAB9A P51151 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
NPC1 O15118 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MAPT P10636 1/20 0.45
G6PD P11413 1/20 0.45
PKM P14618 1/20 0.45
ALOX12 P18054 1/20 0.45
HKDC1 Q2TB90 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PARP1 P09874 2/20 0.43
GABRA1 P14867 2/20 0.43
GABRA5 P31644 2/20 0.43
GABRA3 P34903 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9256388 0.89 ADORA3 (0.55) ADORA2AADORA3POLBKDM4EALDH1A1
SCHEMBL9265209 0.87 POLB (0.48) ADORA1ADORA3POLBKDM4EALDH1A1
SCHEMBL9259533 0.87 MAP4K4 (0.59) ADORA2AADORA3POLBKDM4ERAB9A
SCHEMBL9262896 0.86 ADORA3 (0.49) ADORA3POLBKDM4ERAB9AALDH1A1
SCHEMBL9256089 0.83 ADORA3 (0.54) ADORA2AADORA3POLBKDM4ERAB9A
SCHEMBL9265898 0.81 KDM4E (0.55) ADORA1ADORA2AADORA3KDM4ERAB9A
SCHEMBL9266972 0.81 POLB (0.47) ADORA1ADORA3POLBKDM4ERAB9A
SCHEMBL7269351 0.80 POLB (0.55) ADORA3POLBKDM4EALDH1A1HPGD
SCHEMBL9264849 0.79 MAP4K4 (0.54) ADORA1ADORA2AADORA3POLBKDM4E
SCHEMBL9261950 0.79 ADORA3 (0.49) ADORA3POLBKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993004066-A1 CERTAIN IMIDAZOQUINOXALINOLS; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-03-04 WO claimed
US-5182386-A G-Aminobutyric Acid NEUROGEN CORPORATION (US) 1993-01-26 US claimed
WO-1995033735-A1 EPOXYCYCLOPENTANE DERIVATIVES AND THEIR USE AS FRAGRANCES HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) 1995-12-14 WO disclosed
US-5473073-A Useful in diagnosis or treatment of anxiety, sleep and seizure disorders, overdose with bezodiazepine drug and memory enhancement NEUROGEN CORPORATION (US) 1995-12-05 US disclosed
WO-1993004066-A1 CERTAIN IMIDAZOQUINOXALINOLS; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-03-04 WO disclosed
US-5182386-A G-Aminobutyric Acid NEUROGEN CORPORATION (US) 1993-01-26 US disclosed