SCHEMBL9259828

SCHEMBL9259828

Cc1cc(=O)c(-c2ccc(C(F)(F)F)cc2)c(C)o1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.61
MAPT P10636 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP4B1 P13584 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP3A5 P20815 1/20 0.42
CYP2A7 P20853 1/20 0.42
CYP3A7 P24462 1/20 0.42
CYP2F1 P24903 1/20 0.42
CYP2C18 P33260 1/20 0.42
CYP2C19 P33261 1/20 0.42
CYP2J2 P51589 1/20 0.42
CYP4F2 P78329 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9268345 0.92 PTGS2 (0.55) PTGS2MAPTCYP1A1CYP1A2CYP2E1
SCHEMBL13761581 0.85 PTGS2 (0.48) PTGS2MAPTCYP1A1CYP1A2CYP2E1
SCHEMBL9266616 0.84 PTGS2 (0.49) PTGS2
SCHEMBL9271064 0.81 PTGS2 (0.58) PTGS2MAPTMAOB
SCHEMBL9271388 0.80 PTGS2 (0.45) PTGS2MAPTAR
SCHEMBL9264074 0.80 LMNA (0.49) PTGS2MAPT
SCHEMBL9267689 0.80 PTGS2 (0.57) PTGS2MAPTMAOB
SCHEMBL4468876 0.79 PTGS2 (0.43) PTGS2MAOB
SCHEMBL3394581 0.78 PTGS2 (0.58) PTGS2
SCHEMBL9263874 0.78 PTGS2 (0.58) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403934-A Heterocyclic compounds BURROUGHS WELLCOME CO. (US) 1995-04-04 US disclosed
WO-1991013873-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-19 WO disclosed
EP-0447164-A1 Heterocyclic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-18 EP disclosed