SCHEMBL9260508

SCHEMBL9260508

CCn1c2ccc(OC)cc2c2c3c(c4c5cc(OC)ccc5[nH]c4c21)C(=O)NC3

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYLK Q15746 5/20 0.76
ROCK2 O75116 5/20 0.62
PDGFRB P09619 1/20 0.49
MAP3K9 P80192 1/20 0.47
DLK1 P80370 1/20 0.47
MAP3K10 Q02779 1/20 0.47
MAP3K11 Q16584 1/20 0.47
KDR P35968 1/20 0.46
TEK Q02763 1/20 0.46
PRKD3 O94806 1/20 0.46
PRKCG P05129 1/20 0.46
PRKCB P05771 1/20 0.46
PRKCA P17252 1/20 0.46
PRKCH P24723 1/20 0.46
PRKCI P41743 1/20 0.46
PRKCE Q02156 1/20 0.46
PRKCQ Q04759 1/20 0.46
PRKCZ Q05513 1/20 0.46
PRKCD Q05655 1/20 0.46
PRKD1 Q15139 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9265479 0.96 MYLK (0.71) MYLKROCK2PDGFRBMAP3K9DLK1
SCHEMBL9254743 0.88 MYLK (0.69) MYLKROCK2MAP3K9MAP3K10MAP3K11
SCHEMBL9544892 0.87 MYLK (0.75) MYLKROCK2MAP3K9DLK1MAP3K10
SCHEMBL9826964 0.87 MYLK (0.59) MYLKROCK2PDGFRBMAP3K9DLK1
SCHEMBL9544881 0.87 MYLK (1.00) MYLKROCK2MAP3K9DLK1MAP3K10
SCHEMBL9544714 0.83 MYLK (0.93) MYLKROCK2MAP3K9DLK1MAP3K10
SCHEMBL9263673 0.82 ROCK2 (0.87) MYLKROCK2PDGFRBMAP3K9MAP3K11
SCHEMBL9195167 0.80 ROCK2 (0.74) MYLKROCK2MAP3K9MAP3K11PRKD3
SCHEMBL9260091 0.77 ROCK2 (0.78) MYLKROCK2PDGFRBMAP3K9MAP3K11
SCHEMBL9263506 0.77 ROCK2 (0.78) MYLKROCK2PDGFRBMAP3K9MAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993024490-A1 USE OF INDOLOCARBAZOLS IN AIDS TREATMENT Gödecke Aktiengesellschaft (DE) 1993-12-09 WO claimed
US-5438050-A Indolocarbazole derivatives, processes for their preparation and compositions containing them GODECKE AKTIENGESELLSCHAFT (DE) 1995-08-01 US disclosed
WO-1993024490-A1 USE OF INDOLOCARBAZOLS IN AIDS TREATMENT Gödecke Aktiengesellschaft (DE) 1993-12-09 WO disclosed
EP-0370236-B1 INDOLOCARBAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS GÖDECKE AKTIENGESELLSCHAFT (DE) 1991-12-27 EP disclosed
EP-0370236-A1 Indolocarbazole derivatives, processes for their preparation and their use as medicaments GÖDECKE AKTIENGESELLSCHAFT (DE) 1990-05-30 EP disclosed