SCHEMBL9260561

SCHEMBL9260561

CCOC(C)n1c(C(=O)C2CCN(C(C)(OC)C(=O)OC)CC2)nc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.39
TACR2 P21452 1/20 0.39
TACR1 P25103 1/20 0.39
KDM4E B2RXH2 2/20 0.35
POLB P06746 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
BLM P54132 1/20 0.34
OPRM1 P35372 3/20 0.33
OPRD1 P41143 3/20 0.33
OPRK1 P41145 3/20 0.33
OGFRL1 Q5TC84 3/20 0.33
PROKR1 Q8TCW9 1/20 0.33
PDE6D O43924 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MCHR1 Q99705 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9267727 0.92 HRH1 (0.39) HRH1TACR2TACR1KDM4EPOLB
SCHEMBL9263400 0.81 STS (0.44) KDM4EOPRM1OPRD1OGFRL1SMN1; SMN2
SCHEMBL9268872 0.80 TACR2 (0.44) HRH1TACR2TACR1KDM4EMEN1
SCHEMBL9258711 0.79 REN (0.40) HRH1TACR2TACR1KDM4EPOLB
SCHEMBL9260703 0.77 HRH1 (0.42) HRH1TACR2TACR1KDM4EHSD17B10
SCHEMBL9258366 0.77 HRH1 (0.63) HRH1TACR2TACR1ALDH1A1
SCHEMBL9261042 0.77 TACR2 (0.66) HRH1TACR2TACR1KDM4EPOLB
Hydrochloric Acid SCHEMBL9259556 0.76 TACR2 (0.65) HRH1TACR2TACR1KDM4EPOLB
SCHEMBL9259439 0.75 STS (0.44) KDM4EKMT2AOPRM1OPRD1OGFRL1
SCHEMBL9268748 0.73 HRH1 (0.41) HRH1TACR2TACR1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US claimed
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed