SCHEMBL9263133

SCHEMBL9263133

OC1(c2ccns2)CCCc2cc(Br)ccc21

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.41
CYP11B2 P19099 5/20 0.41
CYP11B1 P15538 4/20 0.41
CYP17A1 P05093 3/20 0.41
SYK P43405 1/20 0.39
APP P05067 1/20 0.34
BACE1 P56817 1/20 0.34
PARP1 P09874 1/20 0.33
PGR P06401 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8746293 0.84 KDM1A (0.44) CYP3A4CYP11B2CYP11B1CYP17A1BACE1
SCHEMBL8746261 0.81 KDM1A (0.47) CYP3A4CYP11B2CYP11B1CYP17A1SYK
SCHEMBL17028624 0.69 PGR (0.48) CYP3A4CYP11B2CYP11B1CYP17A1SYK
SCHEMBL16198401 0.67 SYK (0.37) CYP3A4CYP11B2CYP11B1CYP17A1SYK
SCHEMBL30558325 0.66 APP (0.39) CYP3A4CYP11B2CYP11B1CYP17A1APP
SCHEMBL17361959 0.66 APP (0.39) CYP3A4CYP11B2CYP11B1CYP17A1APP
SCHEMBL14053361 0.66 APP (0.40) CYP3A4CYP11B2CYP11B1CYP17A1APP
SCHEMBL2016698 0.66 BACE1 (0.43) APPBACE1PARP1
SCHEMBL14053247 0.65 BACE1 (0.38) SYKAPPBACE1PARP1
SCHEMBL13900252 0.65 CYP3A4 (0.45) CYP3A4CYP11B2CYP11B1CYP17A1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378721-A AROMATASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1995-01-03 US disclosed
US-5246952-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1993-09-21 US disclosed
EP-0477141-A1 Heteroarylmethylbenzols aromatase inhibitors CIBA-GEIGY AG (CH) 1992-03-25 EP disclosed