SCHEMBL9265451

SCHEMBL9265451

N#Cc1ccc(Cc2csnc2-c2ccc(C#N)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
LOXL2 Q9Y4K0 2/20 0.40
CYP19A1 P11511 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
NSD2 O96028 1/20 0.38
CYP2A6 P11509 1/20 0.38
LRRK2 Q5S007 1/20 0.37
CDC25A P30304 1/20 0.37
CDC25B P30305 1/20 0.37
CDC25C P30307 1/20 0.37
SAE1 Q9UBE0 1/20 0.36
UBA2 Q9UBT2 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.36
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9263382 0.72 LOXL2 (0.40) CYP11B1CYP11B2LOXL2CYP19A1HRH3
SCHEMBL2354871 0.72 CYP11B2 (0.48) CYP11B1CYP11B2LOXL2CYP19A1HRH3
SCHEMBL14155434 0.71 LOXL2 (0.58) CYP11B2LOXL2CYP19A1HRH3CYP2A6
SCHEMBL16848648 0.71 LOXL2 (0.58) CYP11B2LOXL2CYP19A1HRH3CYP2A6
Hydrochloric Acid SCHEMBL1507784 0.71 CYP11B2 (0.47) CYP11B1CYP11B2LOXL2CYP19A1HRH3
SCHEMBL9790872 0.69 CYP11B2 (0.48) CYP11B1CYP11B2CYP19A1HRH3LRRK2
SCHEMBL1344068 0.69 LOXL2 (0.65) LOXL2CYP19A1HRH3CYP2A6SAE1
SCHEMBL9165264 0.67 CYP11B2 (0.43) CYP11B1CYP11B2CYP19A1NSD2GAA
SCHEMBL2352121 0.66 CYP11B1 (0.45) CYP11B1CYP11B2LOXL2CYP19A1HRH3
SCHEMBL2356830 0.64 CYP11B1 (0.43) CYP11B1CYP11B2LOXL2CYP19A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378721-A AROMATASE INHIBITORS CIBA-GEIGY CORPORATION (US) 1995-01-03 US disclosed
US-5246952-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1993-09-21 US disclosed