SCHEMBL9267190

SCHEMBL9267190

Fc1ccc2ncn3ncnc3c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
USP10 Q14694 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.37
USP13 Q92995 1/20 0.37
HTT P42858 3/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HCRTR1 O43613 1/20 0.35
MAP4K4 O95819 2/20 0.34
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29648618 0.75 KDM4E (0.49) HTTMEN1KMT2AALDH1A1KDM4E
SCHEMBL30393692 0.71 LMNA (0.43) MAP4K4MAPT
SCHEMBL30277469 0.70 MAOB (0.50) PARP1ALDH1A1KDM4EGABRG2GABRB3
SCHEMBL29790789 0.67 EGFR (0.42) HTTMEN1KMT2AALDH1A1KDM4E
SCHEMBL9919060 0.64 L3MBTL1 (0.59) PARP1ALDH1A1KDM4EL3MBTL1
SCHEMBL28674308 0.62 USP10 (0.45) PARP1CCNCCDK8USP10PIK3C3
SCHEMBL30106860 0.62 PRKCI (0.42)
SCHEMBL19161108 0.62 USP10 (0.49) PARP1CCNCCDK8USP10PIK3C3
SCHEMBL18312194 0.62 MAP4K4 (0.74) MAP4K4
SCHEMBL3737053 0.62 HTT (0.49) PARP1CCNCCDK8USP10PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed
EP-0519307-A2 Tetracyclic Imidazodiazepines F. HOFFMANN-LA ROCHE AG (CH) 1992-12-23 EP disclosed