SCHEMBL9275609

SCHEMBL9275609

N=C(N)NCCC[C@H](C(=O)O)N(Cc1ccncc1)C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
LMNA P02545 2/20 0.38
TSHR P16473 2/20 0.38
MEN1 O00255 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
MAPT P10636 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
HSD17B10 Q99714 1/20 0.38
F10 P00742 1/20 0.37
EPHX2 P34913 2/20 0.37
ACKR3 P25106 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112682 0.94 CYP2C9 (0.38) CYP2C9CYP2C19LMNATSHRMEN1
SCHEMBL9200838 0.90 CNR1 (0.42) MEN1KMT2ACNR1CNR2TDP1
SCHEMBL9195693 0.89 NPY1R (0.42) CNR1CNR2TDP1
SCHEMBL9199526 0.88 CNR1 (0.43) LMNAMAPTCNR1CNR2TDP1
SCHEMBL9201122 0.88 TDP1 (0.48) CYP2C9CYP2C19LMNAMEN1KMT2A
SCHEMBL9196217 0.88 MEN1 (0.42) MEN1KMT2AF10CNR1CNR2
SCHEMBL30905434 0.86 CNR1 (0.41) MEN1KMT2AF10CNR1CNR2
SCHEMBL1389118 0.86 CNR1 (0.41) MEN1KMT2AF10CNR1CNR2
SCHEMBL9195083 0.85 CNR1 (0.43) KMT2AACKR3CNR1CNR2TDP1
SCHEMBL9194746 0.85 CNR1 (0.43) KMT2AACKR3CNR1CNR2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680469-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME Dr. Karl Thomae GmbH (DE) 1995-11-08 EP disclosed
WO-1994017035-A1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME DR. KARL THOMAE GMBH (DE) 1994-08-04 WO disclosed