SCHEMBL9280474

SCHEMBL9280474

O=C(O)c1nc(S)[nH]c1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 8/20 0.48
CYP1A2 P05177 1/20 0.48
MAPK1 P28482 1/20 0.48
CASP1 P29466 1/20 0.48
CYP2C19 P33261 1/20 0.48
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LDHA P00338 1/20 0.31
LDHB P07195 1/20 0.31
LMNA P02545 2/20 0.30
RNASEH1 O60930 1/20 0.30
ERCC1 P07992 1/20 0.30
FEN1 P39748 1/20 0.30
ERCC4 Q92889 1/20 0.30
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIK1 P39086 1/20 0.30
GRIA1 P42261 1/20 0.30
GRIA2 P42262 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9232538 0.76 PIN1 (0.50) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL11475671 0.74 PIN1 (0.50) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL28169947 0.74 PIN1 (0.50) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL2522013 0.73 PIN1 (0.48) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL213561 0.73 PIN1 (0.48) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL10403221 0.73 PIN1 (0.48) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL2811194 0.73 PIN1 (0.48) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL11008167 0.72 PIN1 (0.44) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL11491730 0.71 PIN1 (0.47) PIN1CYP1A2MAPK1CASP1CYP2C19
SCHEMBL5762937 0.69 PIN1 (0.49) PIN1CYP1A2MAPK1CASP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-60016992-A None JP disclosed
EP-0313724-B1 Bis (acyloxymethyl) imidazole Derivative UNIV NEW YORK STATE RES FOUND (US) 1995-08-09 EP disclosed
CN-1021910-C LANKACIDIN DERIVATIVES AND PRODUCTION THEREOF TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-08-25 CN disclosed
US-4914206-A ANTIBIOTICS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-04-03 US disclosed
EP-0226896-A2 Lankacidin derivatives and production thereof Takeda Chemical Industries, Ltd. (JP) 1987-07-01 EP disclosed
EP-0132501-A2 Cephalosporin derivatives, their preparation and pharmaceutical compositions AJINOMOTO CO., INC. (JP) 1985-02-13 EP disclosed
JP-S6016992-A IMIDAZOLEDICARBOXYLIC ACID DERIVATIVE, ITS PREPARATION AND ITS USE AJINOMOTO CO INC 1985-01-28 JP disclosed
US-4217450-A ANTIBIOTICS, BACTERICIDES AJINOMOTO COMPANY, INCORPORATED (JP) 1980-08-12 US disclosed