SCHEMBL9283240

SCHEMBL9283240

NCN1C(=O)CC[C@@H](c2ccccc2)[C@@H]1c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.53
MDM2 Q00987 6/20 0.53
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
POLB P06746 1/20 0.45
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
SRD5A1 P18405 1/20 0.40
HTT P42858 1/20 0.39
HTR2C P28335 7/20 0.39
HTR2B P41595 6/20 0.39
HTR2A P28223 4/20 0.39
MAOB P27338 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9283243 1.00 TP53 (0.53) TP53MDM2MEN1KMT2APOLB
SCHEMBL9283247 1.00 TP53 (0.53) TP53MDM2MEN1KMT2APOLB
SCHEMBL9309239 0.84 TP53 (0.53) TP53MDM2MEN1KMT2APOLB
SCHEMBL9309243 0.84 TP53 (0.53) TP53MDM2MEN1KMT2APOLB
SCHEMBL9309234 0.84 TP53 (0.53) TP53MDM2MEN1KMT2APOLB
SCHEMBL11477337 0.79 CHRM2 (0.57) TP53MDM2MEN1KMT2APOLB
SCHEMBL21104990 0.69 KMT2A (0.51) TP53MDM2MEN1KMT2APOLB
SCHEMBL19750826 0.68 SIGMAR1 (0.45) TP53MDM2MEN1KMT2APOLB
SCHEMBL21056614 0.66 KMT2A (0.76) MEN1KMT2APOLBSRD5A1HTT
SCHEMBL25017953 0.66 CHRM2 (0.57) MEN1KMT2APOLBCHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995023135-A1 DIPHENYL-2-PIPERIDINONE AND -2-PYRROLIDINONE DERIVATIVES HAVING ANTI-CONVULSANT AND NEUROPROTECTIVE ACTIVITY FISONS CORPORATION (US) 1995-08-31 WO claimed
US-5334720-A Diphenyl-1-(aminoalkyl)-2-piperidinone and -2-pyrrolidinone derivatives having anticonvulsant properties FISONS CORPORATION (US) 1994-08-02 US disclosed