SCHEMBL9286154

SCHEMBL9286154

CCCC[Si](C)(C)Nc1nc(Cl)c2cc[nH]c2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 5/20 0.34
JAK2 O60674 5/20 0.34
PAK4 O96013 5/20 0.34
RET P07949 5/20 0.34
LTK P29376 5/20 0.34
KDR P35968 5/20 0.34
MAPK8 P45983 5/20 0.34
MAPK9 P45984 5/20 0.34
RPS6KA3 P51812 5/20 0.34
JAK3 P52333 5/20 0.34
MAP2K1 Q02750 5/20 0.34
MST1R Q04912 5/20 0.34
PTK2 Q05397 5/20 0.34
MAP4K2 Q12851 5/20 0.34
ROCK1 Q13464 5/20 0.34
LRRK2 Q5S007 5/20 0.34
AURKB Q96GD4 5/20 0.34
CLK4 Q9HAZ1 5/20 0.34
ALK Q9UM73 5/20 0.34
DAPK3 O43293 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8907430 0.74 AXL (0.34) AURKAJAK2PAK4RETLTK
SCHEMBL16743055 0.73 TYRO3 (0.40) AURKAJAK2PAK4RETLTK
SCHEMBL9280468 0.72 HRH4 (0.34) LRRK2ADORA2AADORA1
SCHEMBL15720119 0.69 KCNH3 (0.41) AURKAJAK2PAK4RETLTK
SCHEMBL15557725 0.68 PRKCI (0.39) AURKAJAK2PAK4RETLTK
SCHEMBL4734624 0.66 RAD52 (0.45) JAK2JAK1KMT2A
SCHEMBL691603 0.65 PRKCI (0.44) JAK2PAK4RETLTKKDR
SCHEMBL29700716 0.65 PRKCI (0.44) JAK2PAK4RETLTKKDR
SCHEMBL311465 0.64 MEN1 (0.47) KDRJAK1ADORA2AADORA1PDGFRB
SCHEMBL13666508 0.62 PRKCI (0.41) JAK2DYRK1AJAK1AXLPRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646423-A1 NOVEL COMPOUNDS AS RESPIRATORY STIMULANTS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES Galleon Pharmaceuticals, Inc. (US) 2013-10-09 EP disclosed
WO-2012074999-A1 NOVEL COMPOUNDS AS RESPIRATORY STIMULANTS FOR TREATMENT OF BREATHING CONTROL DISORDERS OR DISEASES GALLEON PHARMACEUTICALS, INC. (US) 2012-06-07 WO disclosed