SCHEMBL9286203

SCHEMBL9286203

COc1cccc2c1CC(CCCNCCCCN1C(=O)c3ccccc3S1(=O)=O)CC2

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.54
DRD2 P14416 5/20 0.51
DRD4 P21917 1/20 0.51
DRD5 P21918 1/20 0.51
DRD3 P35462 1/20 0.51
HTR2A P28223 3/20 0.51
HTR7 P34969 3/20 0.51
HTR6 P50406 3/20 0.51
ACHE P22303 1/20 0.48
CA12 O43570 3/20 0.44
CA9 Q16790 2/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ELANE P08246 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8971218 0.92 HTR1A (0.59) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL9674186 0.85 HTR1A (0.55) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL8996726 0.84 HTR1A (0.49) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL8970423 0.84 HTR1A (0.53) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL8970224 0.79 HTR1A (0.72) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL8971004 0.77 HTR1A (0.75) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL7935857 0.77 HTR1A (0.57) HTR1ADRD2DRD4DRD5DRD3
Hydrochloric Acid SCHEMBL9243980 0.77 HTR1A (0.56) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL7926512 0.77 HTR1A (0.56) HTR1ADRD2DRD4DRD5DRD3
SCHEMBL8970653 0.77 HTR1A (0.41) HTR1ADRD2DRD4DRD5DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463105-A Therapy for cardiovascular, nervous system disorders BAYER AKTIENGESELLSCHAFT (DE) 1995-10-31 US disclosed
US-5298513-A Serotonin antagonist BAYER AKTIENGESELLSCHAFT (DE) 1994-03-29 US disclosed
US-5026857-A Cetnral nervous system disorders; antiserotonine agent BAYER AKTIENGESELLSCHAFT (DE) 1991-06-25 US disclosed
US-4880802-A CENTRAL NERVOUS SYSTEM BAYER AKTIENGESELLSCHAFT (DE) 1989-11-14 US disclosed