SCHEMBL9289357

SCHEMBL9289357

CNC(=O)c1cc(Cl)cc(Cl)c1NC(=O)C1CC(Br)=NN1c1ncccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 12/20 0.39
TRPV1 Q8NER1 1/20 0.34
EPHX2 P34913 1/20 0.34
PHGDH O43175 1/20 0.34
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1148395 0.93 MALT1 (0.43) MALT1PHGDHDHODH
SCHEMBL9290052 0.91 MALT1 (0.37) MALT1
SCHEMBL13884579 0.91 MALT1 (0.39) MALT1TRPV1PHGDHDHODH
SCHEMBL9290207 0.91 MALT1 (0.40) MALT1TRPV1EPHX2
SCHEMBL13961540 0.90 MALT1 (0.41) MALT1TRPV1EPHX2PHGDH
SCHEMBL11888068 0.90 MALT1 (0.41) MALT1TRPV1EPHX2
SCHEMBL9290241 0.88 MALT1 (0.41) MALT1TRPV1PHGDHDHODH
SCHEMBL9290202 0.87 MALT1 (0.37) MALT1TRPV1EPHX2
SCHEMBL12438369 0.86 MALT1 (0.40) MALT1TRPV1PHGDHDHODH
SCHEMBL13002825 0.86 MALT1 (0.40) MALT1TRPV1PHGDHDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012092827-A1 CHEMICAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2012-07-12 WO disclosed
WO-2012069008-A1 3-SUBSTITUTED SPIROHETEROCYCLIC FURAN AND THIOFURAN DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-31 WO disclosed
WO-2011113756-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-09-22 WO disclosed
WO-2011095462-A1 INSECTICIDAL COMPOUNDS SYNGENTA PARTICIPATIONS AG (CH) 2011-08-11 WO disclosed
EP-2332411-A1 Fungicidal compositions Syngenta Participations AG (CH) 2011-06-15 EP disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067203-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067131-A1 SPIROHETEROCYCLIC DIONE DERIVATIVES USED AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
EP-2213167-A1 Anthranilamide derivatives and their use for the control of insects and acari Syngenta Participations AG (CH) 2010-08-04 EP disclosed
WO-2010066780-A1 SPIROHETEROCYCLIC N-OXYPIPERIDINES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-17 WO disclosed
WO-2010063670-A1 SPIROHETEROCYCLIC N-OXYAMIDES AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2010-06-10 WO disclosed
WO-2009024341-A2 CONDENSED ANTHRAN I LAMI DE DERIVATIVES AS INSECTISIDES SYNGENTA PARTICIPATIONS AG, (CH) 2009-02-26 WO disclosed
WO-2009010260-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-01-22 WO disclosed