SCHEMBL9290202

SCHEMBL9290202

CNC(=O)c1cc(Cl)cc(Cl)c1NC(=O)C1CC(C(F)(F)F)=NN1c1ncccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 12/20 0.37
TRPV1 Q8NER1 3/20 0.37
RBP4 P02753 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9290237 0.93 MALT1 (0.41) MALT1TRPV1RBP4LMNAPOLB
SCHEMBL12294895 0.91 MALT1 (0.38) MALT1TRPV1RBP4
SCHEMBL9289364 0.91 MALT1 (0.36) MALT1TRPV1RBP4
SCHEMBL9290207 0.89 MALT1 (0.40) MALT1TRPV1RBP4EPHX2
SCHEMBL13356445 0.88 ALDH1A1 (0.34) MALT1TRPV1RBP4
SCHEMBL11888068 0.88 MALT1 (0.41) MALT1TRPV1EPHX2
SCHEMBL13961540 0.88 MALT1 (0.41) MALT1TRPV1EPHX2
SCHEMBL9289357 0.87 MALT1 (0.39) MALT1TRPV1EPHX2
SCHEMBL9290200 0.87 MALT1 (0.39) MALT1TRPV1RBP4LMNAPOLB
SCHEMBL9290246 0.87 MALT1 (0.39) MALT1TRPV1RBP4LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197844-B1 SPIROHETEROCYCLIC PYRROLIDINE DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-07-25 EP disclosed
WO-2012069008-A1 3-SUBSTITUTED SPIROHETEROCYCLIC FURAN AND THIOFURAN DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-05-31 WO disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2009049851-A1 SPIROHETEROCYCLIC PYRROLIDINE DIONE DERIVATIVES USEFUL AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-04-23 WO disclosed
WO-2009024341-A2 CONDENSED ANTHRAN I LAMI DE DERIVATIVES AS INSECTISIDES SYNGENTA PARTICIPATIONS AG, (CH) 2009-02-26 WO disclosed
WO-2009021717-A2 PESTICIDAL FORMULATION SYNGENTA PARTICIPATIONS AG (CH) 2009-02-19 WO disclosed
WO-2009010260-A2 CONDENSED ANTHRANILAMIDE INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2009-01-22 WO disclosed
WO-2008064891-A1 N-CYANOALKYLANTHRANILAMIDES AS INSECTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2008-06-05 WO disclosed