SCHEMBL928982

SCHEMBL928982

N#Cc1cc(N2C[C@H]3CN(C(=O)OCc4ccccc4)C[C@H]32)cnc1-c1cccs1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 7/20 0.39
HCRTR2 O43614 7/20 0.39
GRIN2B Q13224 3/20 0.38
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
TGM1 P22735 1/20 0.37
CYP2C9 P11712 2/20 0.36
CYP2D6 P10635 1/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
CHRM4 P08173 1/20 0.35
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1795535 0.86 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL929833 0.84 CHRNB2 (0.49) GRIN2BF13A1TGM2TGM1CYP2C9
SCHEMBL654606 0.78 CHRNB2 (0.47) F13A1TGM2TGM1ALDH1A1HPGD
SCHEMBL649574 0.78 CHRNB2 (0.47) F13A1TGM2TGM1ALDH1A1HPGD
Fumaric Acid SCHEMBL929017 0.77 HRH3 (0.38) HCRTR1HCRTR2ALDH1A1HPGDMEN1
Fumaric Acid SCHEMBL929018 0.77 HRH3 (0.38) HCRTR1HCRTR2ALDH1A1HPGDMEN1
Fumaric Acid SCHEMBL929016 0.77 HRH3 (0.38) HCRTR1HCRTR2ALDH1A1HPGDMEN1
SCHEMBL930264 0.77 HRH3 (0.44) HCRTR1HCRTR2
SCHEMBL3295704 0.75 KDM4E (0.45) GRIN2BF13A1TGM2TGM1CYP2C9
SCHEMBL654459 0.75 CHRNB2 (0.45) GRIN2BF13A1TGM2TGM1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872010-B2 Substituted diazabicycloalkane derivatives having affinity for nicotinic acetylcholine receptors ABBOTT LABORATORIES (US) 2011-01-18 US disclosed