SCHEMBL9290394

SCHEMBL9290394

CCn1c(N(C)CC(C)N)nc2c1c(=O)n(Cc1cn3c(C)cccc3n1)c(=O)n2C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.40
ADORA1 P30542 2/20 0.40
MAPT P10636 3/20 0.35
ADORA2A P29274 1/20 0.35
ALDH1A1 P00352 5/20 0.35
TSHR P16473 3/20 0.35
MAPK1 P28482 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
HPGD P15428 1/20 0.33
ATM Q13315 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
RAB9A P51151 2/20 0.33
DCTPP1 Q9H773 1/20 0.33
GFER P55789 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8271562 0.90 DPP4 (0.39) ADORA3ADORA1
SCHEMBL13954990 0.87 ADORA3 (0.39) ADORA3ADORA1MAPTADORA2AALDH1A1
SCHEMBL9290387 0.80 ALDH1A1 (0.42) ADORA3ADORA1MAPTALDH1A1TSHR
SCHEMBL13954926 0.79 DPP4 (0.39) ADORA3ADORA1MAPTALDH1A1TSHR
SCHEMBL13955116 0.78 HSD17B10 (0.42) MAPTALDH1A1TSHRMAPK1NPSR1
SCHEMBL8271557 0.78 DPP4 (0.42) ADORA3ADORA1
SCHEMBL10030473 0.77 DPP4 (0.50) ADORA3MAPTALDH1A1TSHRMAPK1
SCHEMBL13954913 0.77 DPP4 (0.50) ADORA3MAPTALDH1A1TSHRMAPK1
SCHEMBL13955070 0.76 DPP4 (0.49) ADORA3ADORA1MAPTALDH1A1TSHR
SCHEMBL8272349 0.76 DPP4 (0.48) ADORA3ADORA1MAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797093-B1 NOVEL 3-METHYL-7-BUTINYL-XANTHINES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP disclosed
US-7495002-B2 3-methyl-7-butinyl-xanthines, the preparation thereof and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-24 US disclosed