SCHEMBL9290709

SCHEMBL9290709

C=C(C)c1nc(N)nc(C)c1C#N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.39
ALDH1A1 P00352 9/20 0.36
HPGD P15428 6/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 5/20 0.35
CYP1A2 P05177 1/20 0.35
ADORA1 P30542 5/20 0.34
ADORA2A P29274 4/20 0.34
HSD17B10 Q99714 5/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
CASP1 P29466 1/20 0.32
RAB9A P51151 1/20 0.32
CASP7 P55210 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 2/20 0.31
ADRA2A P08913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9288685 0.78 ALDH1A1 (0.43) LMNAALDH1A1HPGDGAAKDM4E
SCHEMBL17342569 0.72 ALDH1A1 (0.48) ALDH1A1HPGDGAAKDM4EADORA1
SCHEMBL14310461 0.71 LMNA (0.46) LMNAALDH1A1HPGDGAAKDM4E
SCHEMBL31575894 0.69 ALDH1A1 (0.55) ALDH1A1HPGDGAAKDM4EADORA1
SCHEMBL17401071 0.69 ADORA1 (0.38) LMNAALDH1A1HPGDGAAKDM4E
SCHEMBL11900926 0.69 ALDH1A1 (0.55) ALDH1A1HPGDGAAKDM4EADORA1
SCHEMBL18300545 0.69 KDM4E (0.39) ALDH1A1HPGDGAAKDM4EADORA1
SCHEMBL9289563 0.68 LMNA (0.52) LMNAALDH1A1HPGDGAAKDM4E
SCHEMBL18868083 0.67 HTT (0.37) LMNAALDH1A1HPGDGAAKDM4E
SCHEMBL15429586 0.67 ALDH1A1 (0.37) LMNAALDH1A1HPGDGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071501-A1 BENZOXAZEPINES ASN INHIBITORS OF P13K/M TOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed