SCHEMBL9292136

SCHEMBL9292136

CC(C)c1cccc(NC(=O)N(C)C)c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.56
FADS1 O60427 1/20 0.55
APEX1 P27695 1/20 0.54
PNPLA2 Q96AD5 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
CA2 P00918 1/20 0.52
MTOR P42345 1/20 0.51
GRIN2D O15399 1/20 0.50
GRIN3B O60391 1/20 0.50
GRIN1 Q05586 1/20 0.50
GRIN2A Q12879 1/20 0.50
GRIN2B Q13224 1/20 0.50
GRIN2C Q14957 1/20 0.50
GRIN3A Q8TCU5 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
NPY5R Q15761 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11716429 0.87 APEX1 (0.55) TP53APEX1PNPLA2HDAC6MEN1
SCHEMBL11409020 0.84 MEN1 (0.55) FADS1MEN1KMT2ACA2MTOR
SCHEMBL19019393 0.84 TP53 (0.69) TP53APEX1PNPLA2HDAC6
SCHEMBL11163949 0.83 TP53 (0.50) TP53APEX1PNPLA2HDAC6MEN1
SCHEMBL7634431 0.83 TP53 (0.56) TP53APEX1PNPLA2HDAC6MEN1
SCHEMBL104492 0.81 ALDH1A1 (0.59) TP53FADS1MEN1KMT2ACA2
SCHEMBL2096083 0.81 FADS1 (0.59) TP53FADS1MEN1KMT2ACA2
SCHEMBL2096086 0.81 FADS1 (0.59) FADS1MEN1KMT2ACA2MTOR
SCHEMBL16980501 0.80 KDM4E (0.51) FADS1MEN1KMT2ACA2GRIN2D
SCHEMBL12569599 0.79 FADS1 (0.61) FADS1MEN1KMT2ACA2GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312576-A1 4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-3,6-DIHYDROPYRIDINE-1-(2H)-CARBOXAMIDE DERIVATIVES AS LIMK AND/OR ROCK KINASES INHIBITORS FOR USE IN THE TREATMENT OF CANCER UNIVERSITÉ DE TOURS (FR) 2023-10-05 US disclosed
US-5321000-A Benzhydryl compounds as herbicide antidotes MONSANTO COMPANY (US) 1994-06-14 US disclosed
US-5162537-A To safen acetamide herbicids used to control grassy and broadleaf weeds in rice, sorghum and wheat MONSANTO COMPANY (US) 1992-11-10 US disclosed
US-4964893-A REDUCING INJURY TO A CROP PLANT MONSANTO COMPANY (US) 1990-10-23 US disclosed
US-4740236-A N-sulfonyl-imino-thiocarbonic acid diesters as herbicide antagonists for the protection of rice crops CIBA-GEIGY CORPORATION (US) 1988-04-26 US disclosed
US-4674229-A SEEDS COATED WITH PLANT SAFENING AGENT CIBA-GEIGY CORPORATION (US) 1987-06-23 US disclosed
US-4648896-A PLANT SAFENING AGENTS CIBA-GEIGY CORPORATION (US) 1987-03-10 US disclosed
US-4493726-A PLANT SAFENING AGENT CIBA GEIGY CORPORATION (US) 1985-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230312576-A1 4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)-3,6-DIHYDROPYRIDINE-1-(2H)-CARBOXAMIDE DERIVATIVES AS LIMK AND/OR ROCK KINASES INHIBITORS FOR USE IN THE TREATMENT OF CANCER LIMK1, LIMK2, ROCK1 TP53 2381/4885FADS1 3683/4885APEX1 2442/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.