SCHEMBL9296265

SCHEMBL9296265

ClCSc1ccccc1Br

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.52
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
LMNA P02545 2/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
PDE7A Q13946 4/20 0.35
PDE7B Q9NP56 2/20 0.34
ALDH1A1 P00352 2/20 0.33
TAAR1 Q96RJ0 1/20 0.32
RAB9A P51151 2/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31378718 1.00 HTR7 (0.52) HTR7MAOAMAOBLMNACA1
SCHEMBL7974171 0.82 MEN1 (0.37) HTR7MAOAMAOBLMNAALDH1A1
SCHEMBL13508978 0.80 HTR7 (0.67) HTR7MAOAMAOBLMNACA1
SCHEMBL5663275 0.79 HTR7 (0.55) HTR7MAOAMAOBLMNACA1
SCHEMBL28754182 0.76 HTR7 (0.52) HTR7MAOAMAOBLMNACA1
SCHEMBL14460773 0.76 HTR7 (0.62) HTR7MAOAMAOBLMNACA1
SCHEMBL1802193 0.76 HTR7 (0.57) HTR7MAOAMAOBLMNACA1
SCHEMBL8779744 0.75 HTR7 (0.32) HTR7MAOAMAOBALDH1A1TAAR1
SCHEMBL28941890 0.74 MEN1 (0.36) HTR7MAOAMAOBCA1CA2
SCHEMBL4334230 0.73 POLB (0.61) HTR7MAOAMAOBLMNACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276053-A Dibenzothiopyranylamines WARNER-LAMBERT COMPANY (US) 1994-01-04 US disclosed
US-5180736-A Treatment and prevention of brain disorders WARNER-LAMBERT COMPANY (US) 1993-01-19 US disclosed
US-5071853-A Amine-substituted hexahydroindeno(2,1-b)pyrroles, -indeno(2,1-c)pyridines or -indeno(2,1-d)azepines; cerebral ischemia or infarction WARNER-LAMBERT COMPANY 1991-12-10 US disclosed
EP-0388977-A2 Polycyclic amines useful as cerebrovascular agents WARNER-LAMBERT COMPANY (US) 1990-09-26 EP disclosed
US-4062846-A CNS STIMULANTS, MUSCLE RELAXANT E. R. SQUIBB & SONS, INC. (US) 1977-12-13 US disclosed
US-3995042-A MUSCLE RELAXANTS, CENTRAL NERVOUS SYSTEM STIMULANTS E. R. SQUIBB & SONS, INC. (US) 1976-11-30 US disclosed
US-3981886-A Amino-benzimidazole derivatives E. R. SQUIBB & SONS, INC. (US) 1976-09-21 US disclosed
US-3966733-A CENTRAL NERVOUS SYSTEM STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1976-06-29 US disclosed
US-3957799-A STIMULANTS, MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1976-05-18 US disclosed
US-3946025-A MUSCLE RELAXANTS E. R. SQUIBB & SONS, INC. (US) 1976-03-23 US disclosed