SCHEMBL9296428

SCHEMBL9296428

CCOC(=O)C1=CCOc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
TSHR P16473 2/20 0.45
MAPT P10636 4/20 0.44
GLA P06280 2/20 0.44
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
CTDSP1 Q9GZU7 2/20 0.41
APAF1 O14727 1/20 0.40
MITF O75030 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TP53 P04637 2/20 0.40
POLB P06746 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5848267 0.83 TSHR (0.47) ALDH1A1TSHRMAPTGLAMEN1
SCHEMBL28812405 0.79 ALDH1A1 (0.39) ALDH1A1TSHRMAPTGLAMEN1
SCHEMBL12764795 0.78 TSHR (0.44) ALDH1A1TSHRMAPTMEN1KMT2A
SCHEMBL17107518 0.78 ATM (0.39) TSHRMAPTMEN1KMT2ALMNA
SCHEMBL9245714 0.77 ALDH1A1 (0.43) ALDH1A1TSHRGLALMNAHSD17B10
SCHEMBL19985040 0.77 SMN1; SMN2 (0.39) ALDH1A1TSHRMAPTGLASMN1; SMN2
SCHEMBL7487263 0.75 ALDH1A1 (0.47) ALDH1A1TSHRMAPTGLAMEN1
SCHEMBL6369076 0.74 NOTUM (0.42) ALDH1A1TSHRMAPTGLAMEN1
SCHEMBL4018002 0.74 TSHR (0.49) ALDH1A1TSHRMAPTMEN1KMT2A
SCHEMBL30255072 0.73 TSHR (0.39) ALDH1A1TSHRMAPTGLAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276053-A Dibenzothiopyranylamines WARNER-LAMBERT COMPANY (US) 1994-01-04 US disclosed
US-5180736-A Treatment and prevention of brain disorders WARNER-LAMBERT COMPANY (US) 1993-01-19 US disclosed
US-5071853-A Amine-substituted hexahydroindeno(2,1-b)pyrroles, -indeno(2,1-c)pyridines or -indeno(2,1-d)azepines; cerebral ischemia or infarction WARNER-LAMBERT COMPANY 1991-12-10 US disclosed
EP-0388977-A2 Polycyclic amines useful as cerebrovascular agents WARNER-LAMBERT COMPANY (US) 1990-09-26 EP disclosed