SCHEMBL9299014

SCHEMBL9299014

O=C(O)[C@@H](Nc1ccccc1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
MDM2 Q00987 2/20 0.49
S1PR3 Q99500 2/20 0.44
S1PR4 O95977 1/20 0.44
S1PR1 P21453 1/20 0.44
S1PR5 Q9H228 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FPR2 P25090 1/20 0.42
SLC6A2 P23975 4/20 0.41
SLC6A4 P31645 4/20 0.41
SLC6A3 Q01959 4/20 0.41
KCNH2 Q12809 4/20 0.41
CYP3A4 P08684 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299009 1.00 KEAP1 (0.51) KEAP1NFE2L2MDM2S1PR3S1PR4
SCHEMBL7584703 0.85 NPC1 (0.53) KEAP1NFE2L2S1PR3S1PR4NPC1
SCHEMBL5882952 0.83 S1PR3 (0.51) KEAP1NFE2L2MDM2S1PR3S1PR4
SCHEMBL11301777 0.82 CA12 (0.45) MEN1KMT2AFPR2CYP3A4CYP2D6
SCHEMBL5883122 0.82 F7 (0.57) MDM2S1PR3S1PR4S1PR1S1PR5
SCHEMBL2484594 0.81 CNR1 (0.53) MDM2NPC1RAB9AMEN1KMT2A
SCHEMBL9298520 0.81 CNR1 (0.53) MDM2NPC1RAB9AMEN1KMT2A
SCHEMBL11211222 0.81 MEN1 (0.55) KEAP1NFE2L2NPC1RAB9AMEN1
SCHEMBL9298095 0.81 KEAP1 (0.52) KEAP1NFE2L2S1PR3S1PR4S1PR1
SCHEMBL9298091 0.81 KEAP1 (0.52) KEAP1NFE2L2S1PR3S1PR4S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5374656-A Nervous system disorders, gastrointestinal disorders RHONE-POULENC RORER, S.A. (FR) 1994-12-20 US disclosed