SCHEMBL9299149

SCHEMBL9299149

COC(=O)c1cnc(N2CCCCC2)nc1N

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 16/20 0.60
SMN1; SMN2 Q16637 2/20 0.55
POLB P06746 2/20 0.55
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9297364 0.84 POLB (0.56) PTPN11SMN1; SMN2POLBKDM4ENPSR1
SCHEMBL14626136 0.84 MAPT (0.56) PTPN11SMN1; SMN2POLBKDM4ENPC1
SCHEMBL27316944 0.83 POLB (0.55) PTPN11SMN1; SMN2POLBKDM4EALDH1A1
SCHEMBL9048339 0.80 POLB (0.51) PTPN11SMN1; SMN2POLBKDM4ENPSR1
SCHEMBL9051143 0.80 POLB (0.51) PTPN11SMN1; SMN2POLBKDM4ENPSR1
SCHEMBL15341329 0.76 MAPT (0.53) SMN1; SMN2POLBKDM4ENPC1RAB9A
SCHEMBL10324214 0.75 POLB (0.45) SMN1; SMN2POLBKDM4ENPC1RAB9A
SCHEMBL23370098 0.74 MAPT (0.54) SMN1; SMN2POLBKDM4ENPC1RAB9A
SCHEMBL10322693 0.74 PTPN11 (0.56) PTPN11SMN1; SMN2POLBKDM4ENPC1
SCHEMBL30468126 0.74 TSHR (0.47) SMN1; SMN2KDM4ENPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305184-B1 Pyrimidines or their pharmaceutically acceptable salts thereof MITSUI PHARMACEUTICALS (JP) 1994-04-27 EP disclosed
US-5304555-A Pyrimidines and pharmaceutically acceptable salts thereof useful in treatment of neurological disorders MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1994-04-19 US disclosed
WO-1989001938-A1 PYRIMIDINES AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF MITSUI PHARMACEUTICALS, INC. (JP) 1989-03-09 WO disclosed