SCHEMBL9299531

SCHEMBL9299531

CC(NC(=O)c1ccccc1)[C@@H](O)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.61
ADRA1A P35348 1/20 0.61
RGS12 O14924 1/20 0.61
GLA P06280 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
PKM P14618 1/20 0.61
ALOX15 P16050 1/20 0.61
TSHR P16473 1/20 0.61
ALOX12 P18054 1/20 0.61
ADRA2C P18825 1/20 0.61
NFKB1 P19838 1/20 0.61
HTR2A P28223 1/20 0.61
CYP2C19 P33261 1/20 0.61
THPO P40225 1/20 0.61
GNAI1 P63096 1/20 0.61
HSD17B10 Q99714 1/20 0.61
KMT2A Q03164 2/20 0.59
MEN1 O00255 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5700232 1.00 CHRM2 (0.61) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL5709299 1.00 CHRM2 (0.61) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL8470684 0.89 CHRM2 (0.53) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL30695641 0.89 UTS2R (0.54) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL8470500 0.85 ALDH1A1 (0.50) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL14828665 0.83 ALDH1A1 (0.53) ALOX15HSD17B10KMT2AMEN1LMNA
SCHEMBL13495008 0.83 ALDH1A1 (0.53) ALOX15HSD17B10KMT2AMEN1LMNA
SCHEMBL16164987 0.83 ADRA2C (0.62) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL14350766 0.81 ADRA2C (0.60) CHRM2ADRA1ARGS12GLACYP3A4
SCHEMBL14393865 0.81 ADRA2C (0.60) CHRM2ADRA1ARGS12GLACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5310911-A Chiral synthesis for producing 1-azabicyclo(2.2.1)heptane-3-carboxylates COTTRELL I F 1994-05-10 US disclosed
US-5124460-A Enantioselective synthesis of 3-substituted 1-azabicyclo (2.2.1)heptanes MERCK SHARP & DOHME LTD. (GB) 1992-06-23 US disclosed
US-5104989-A Chiral synthesis for producing 1-azabicyclo[2.2.1] heptane-3-carboxylates MERCK SHARP & DOHME LTD. (GB) 1992-04-14 US disclosed
EP-0456310-A2 Enantioselective synthesis of 3-substituted 1-azabicyclo [2.2.1]heptanes MERCK SHARP & DOHME LTD. (GB) 1991-11-13 EP disclosed
EP-0398616-A2 Chiral synthesis for producing 1-azabicyclo[2.2.1]heptane-3-carboxylates MERCK SHARP & DOHME LTD. (GB) 1990-11-22 EP disclosed