SCHEMBL9300423

SCHEMBL9300423

CC(C)(C)OC(=O)Nc1ccc(NCC(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.48
PTPN11 Q06124 1/20 0.47
PSMB8 P28062 1/20 0.46
NAMPT P43490 1/20 0.46
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA9 Q16790 1/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
MAPKAPK2 P49137 1/20 0.43
DRD2 P14416 1/20 0.43
MAPK14 Q16539 1/20 0.43
MAP4K4 O95819 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL11643609 0.98 CYP17A1 (0.50) CYP17A1PTGDR2PTPN11PSMB8NAMPT
SCHEMBL18311597 0.85 HDAC1 (0.46) CYP17A1NAMPTCA12CA1CA9
SCHEMBL11649697 0.84 ALDH1A1 (0.40) CYP17A1PTGDR2PTPN11CA12CA1
SCHEMBL13055402 0.84 CYP17A1 (0.59) CYP17A1PTGDR2PTPN11PSMB8NAMPT
SCHEMBL5106835 0.83 CYP17A1 (0.54) CYP17A1PTGDR2PTPN11PSMB8NAMPT
SCHEMBL13193491 0.82 CYP17A1 (0.52) CYP17A1PTGDR2PTPN11PSMB8NAMPT
SCHEMBL14861108 0.82 CYP17A1 (0.52) CYP17A1PTGDR2PTPN11PSMB8NAMPT
SCHEMBL222627 0.82 POLB (0.57) CYP17A1PTGDR2PSMB8NAMPTCA12
SCHEMBL3486818 0.82 NAMPT (0.54) CYP17A1PTGDR2PTPN11NAMPTCA1
SCHEMBL11090977 0.82 NAMPT (0.53) PTPN11NAMPTCA12CA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5362747-A Promoters, inhibitors ABBOTT LABORATORIES (US) 1994-11-08 US disclosed
WO-1994012163-A1 2-NITROARYL AND 2-CYANOARYL COMPOUNDS AS REGULATORS OF NITRIC OXIDE SYNTHASE ABBOTT LABORATORIES (US) 1994-06-09 WO disclosed
US-4111981-A SUBSTITUTED PHENYLGLYCINES SMITHKLINE CORPORATION (US) 1978-09-05 US disclosed
US-4107440-A (CARBOALKOXYALKYLTHIO)-SUBSTITUTED PHENYLGLYCINES SMITHKLINE CORPORATION (US) 1978-08-15 US disclosed
US-4092480-A Intermediates for preparing substituted phenylglycylcephalosporins SMITHKLINE CORPORATION (US) 1978-05-30 US disclosed
US-4044047-A BACTERICIDES SMITHKLINE CORPORATION (US) 1977-08-23 US disclosed
US-4022895-A BACTERICIDE SMITHKLINE CORPORATION (US) 1977-05-10 US disclosed
US-4018921-A BACTERICIDES SMITHKLINE CORPORATION (US) 1977-04-19 US disclosed