SCHEMBL11649697

SCHEMBL11649697

CC(C)(C)OC(=O)NC(=O)CNc1ccc(NCC(=O)O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPT P10636 4/20 0.40
KMT2A Q03164 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
PTPN11 Q06124 1/20 0.39
CYP17A1 P05093 1/20 0.37
CA1 P00915 2/20 0.37
NLRP1 Q9C000 1/20 0.37
CA12 O43570 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA2 P00918 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
AGTR1 P30556 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ERCC1 P07992 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027360 0.89 LMNA (0.48) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL4929584 0.88 MIF (0.44) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL5864432 0.87 ALDH1A1 (0.42) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL11650332 0.86 SMN1; SMN2 (0.44) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL5664612 0.85 ALDH1A1 (0.46) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL11648025 0.85 USP2 (0.42) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL9300423 0.84 CYP17A1 (0.51) ALDH1A1MAPTKMT2ARAB9AMEN1
Water SCHEMBL11643609 0.83 CYP17A1 (0.50) ALDH1A1MAPTKMT2ARAB9AMEN1
SCHEMBL11649700 0.81 SENP1 (0.37) MAPTRAB9APTPN11CYP17A1CA1
SCHEMBL11090977 0.79 NAMPT (0.53) MAPTKMT2AMEN1PTPN11CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4044047-A BACTERICIDES SMITHKLINE CORPORATION (US) 1977-08-23 US claimed
US-4111981-A SUBSTITUTED PHENYLGLYCINES SMITHKLINE CORPORATION (US) 1978-09-05 US disclosed
US-4107440-A (CARBOALKOXYALKYLTHIO)-SUBSTITUTED PHENYLGLYCINES SMITHKLINE CORPORATION (US) 1978-08-15 US disclosed
US-4092480-A Intermediates for preparing substituted phenylglycylcephalosporins SMITHKLINE CORPORATION (US) 1978-05-30 US disclosed
US-4044047-A BACTERICIDES SMITHKLINE CORPORATION (US) 1977-08-23 US disclosed
US-4022895-A BACTERICIDE SMITHKLINE CORPORATION (US) 1977-05-10 US disclosed
US-4018921-A BACTERICIDES SMITHKLINE CORPORATION (US) 1977-04-19 US disclosed
US-4013764-A PHARMACEUTICAL COMPOSITIONS COMPRISING SUBSTITUTED PHENYLGLYCYLCEPHALOSPORINS AND METHODS OF TREATING BACTERIAL INFECTIONS SMITHKLINE CORPORATION (US) 1977-03-22 US disclosed
US-3953439-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-04-27 US disclosed