SCHEMBL9301038

SCHEMBL9301038

COC(=O)c1ccc2c(-c3ccccc3)cc(CO)cc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
EGFR P00533 1/20 0.49
P2RY14 Q15391 1/20 0.48
PTGS2 P35354 1/20 0.47
ALOX5 P09917 1/20 0.46
LCK P06239 1/20 0.45
KIF11 P52732 1/20 0.44
GPR84 Q9NQS5 1/20 0.43
NEK1 Q96PY6 1/20 0.43
SGK1 O00141 1/20 0.43
CAMKK2 Q96RR4 1/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
TSHR P16473 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2926113 0.78 EGFR (0.51) MEN1KMT2AEGFRP2RY14PTGS2
SCHEMBL9300644 0.77 P2RY14 (0.78) P2RY14ALOX5
SCHEMBL29138977 0.76 MEN1 (0.50) MEN1KMT2AEGFRPTGS2LCK
SCHEMBL5776604 0.75 PTPN11 (0.54) LCKCYP4F2CYP4A11CYP19A1CYP11B1
SCHEMBL9303741 0.75 MEN1 (0.52) MEN1KMT2AEGFRPTGS2LCK
SCHEMBL7824090 0.75 EGFR (0.52) MEN1KMT2AEGFRPTGS2SGK1
SCHEMBL9302368 0.74 KDM4E (0.54) MEN1KMT2AP2RY14ALOX5
SCHEMBL3149487 0.74 CYP4A11 (0.50) LCKCYP4F2CYP4A11CYP19A1CYP11B1
SCHEMBL10458005 0.74 PTGS2 (0.76) MEN1KMT2AEGFRPTGS2KIF11
SCHEMBL16502556 0.72 EGFR (0.54) MEN1KMT2AEGFRPTGS2GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1087907-A Heteroaryl naphthalene as white (cell) triolefin biosynthesis inhibitor MERCK FROSST CANADA INC (CA) 1994-06-15 CN disclosed
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed