SCHEMBL9301237

SCHEMBL9301237

Cc1cc2c(cc1C#Cc1cnnc(CC(=O)O)c1)C(C)(C)CCS2

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.41
CYP26A1 O43174 2/20 0.41
RARA P10276 7/20 0.41
RARB P10826 7/20 0.41
RARG P13631 7/20 0.41
KMT2A Q03164 1/20 0.41
RXRA P19793 5/20 0.32
RXRB P28702 3/20 0.32
RXRG P48443 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302684 0.89 RARA (0.46) CYP3A4CYP26A1RARARARBRARG
SCHEMBL9302619 0.88 CYP3A4 (0.39) CYP3A4CYP26A1RARARARBRARG
SCHEMBL9302949 0.85 CYP3A4 (0.57) CYP3A4CYP26A1RARARARBRARG
SCHEMBL6664858 0.84 CYP26A1 (0.46) CYP3A4CYP26A1RARARARBRARG
SCHEMBL6663854 0.82 CYP26A1 (0.47) CYP3A4CYP26A1RARARARBRARG
SCHEMBL6664152 0.82 CYP26A1 (0.45) CYP3A4CYP26A1RARARARBRARG
SCHEMBL9303655 0.82 CYP3A4 (0.43) CYP3A4CYP26A1RARARARBRARG
SCHEMBL9302702 0.81 RARA (0.41) CYP3A4CYP26A1RARARARBRARG
SCHEMBL9302749 0.81 CYP26A1 (0.38) CYP26A1RARARARBRARGRXRA
SCHEMBL9302613 0.80 CYP3A4 (0.39) CYP3A4CYP26A1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed