SCHEMBL9302949

SCHEMBL9302949

CC1(C)CCSc2ccc(C#Cc3cnnc(CC(=O)O)c3)cc21

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.57
CYP26A1 O43174 3/20 0.57
RARB P10826 16/20 0.55
RARG P13631 16/20 0.55
RARA P10276 13/20 0.55
KMT2A Q03164 1/20 0.53
RXRA P19793 3/20 0.40
CRABP2 P29373 1/20 0.39
SSTR5 P35346 1/20 0.34
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303234 0.88 RARB (0.61) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301902 0.88 CYP3A4 (0.53) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301237 0.85 CYP3A4 (0.41) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6666821 0.84 CYP3A4 (0.64) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6665585 0.83 CYP3A4 (0.64) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6664613 0.83 CYP3A4 (0.67) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9302591 0.82 RARB (0.61) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9302103 0.80 RARB (0.56) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9304352 0.80 CYP26A1 (0.46) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9301893 0.79 CYP3A4 (0.52) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed