SCHEMBL9301413

SCHEMBL9301413

N#Cc1ccc2cc(OCc3ccccc3)ccc2c1-c1ccoc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.53
IMPDH2 P12268 1/20 0.48
ALOX5 P09917 7/20 0.46
MAOA P21397 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NSD2 O96028 1/20 0.39
AS3MT Q9HBK9 1/20 0.39
P2RY14 Q15391 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301723 0.79 ALOX5 (0.44) ALOX5
SCHEMBL3648539 0.71 MAOB (1.00) MAOBIMPDH2ALOX5MAOANSD2
SCHEMBL7837193 0.69 MAOB (0.75) MAOBIMPDH2ALOX5MAOANPC1
SCHEMBL3865512 0.69 MAOB (0.77) MAOBIMPDH2ALOX5MAOANSD2
SCHEMBL4260225 0.69 MAOB (0.77) MAOBIMPDH2ALOX5MAOANSD2
SCHEMBL13523861 0.69 MAOB (0.58) MAOBIMPDH2ALOX5MAOANSD2
SCHEMBL13523862 0.68 MAOB (0.57) MAOBIMPDH2ALOX5MAOA
SCHEMBL23887978 0.68 MAOB (0.74) MAOBIMPDH2ALOX5MAOARAB9A
SCHEMBL21124838 0.68 MAOB (0.74) MAOBIMPDH2ALOX5MAOARAB9A
SCHEMBL14677247 0.68 MAOB (0.74) MAOBIMPDH2ALOX5MAOANSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed