SCHEMBL9301446

SCHEMBL9301446

CCc1cc(-c2ccccc2)c2ccc(O)cc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
MEN1 O00255 2/20 0.51
MAPT P10636 2/20 0.51
HPGD P15428 2/20 0.51
KMT2A Q03164 2/20 0.51
MPI P34949 1/20 0.51
ALOX5 P09917 2/20 0.47
ESR2 Q92731 5/20 0.45
CA12 O43570 1/20 0.43
ALDH2 P05091 1/20 0.43
AKR1B1 P15121 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
HSD17B3 P37058 1/20 0.43
SORD Q00796 1/20 0.43
CA9 Q16790 1/20 0.43
ESR1 P03372 4/20 0.42
P2RY14 Q15391 1/20 0.42
CDK4 P11802 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302368 0.87 KDM4E (0.54) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9301150 0.84 KDM4E (0.51) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9300724 0.80 KDM4E (0.46) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL27569906 0.79 KDM4E (0.51) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9301912 0.77 KDM4E (0.46) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9978151 0.76 PTPN1 (0.51) ALDH1A1MAPTHPGDALOX5ESR2
SCHEMBL9302158 0.74 ALDH1A1 (0.50) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL2926113 0.74 EGFR (0.51) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9301722 0.73 P2RY14 (0.63) KDM4EALDH1A1MEN1MAPTHPGD
SCHEMBL9246440 0.73 KDM4E (0.67) KDM4EALDH1A1MEN1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1087907-A Heteroaryl naphthalene as white (cell) triolefin biosynthesis inhibitor MERCK FROSST CANADA INC (CA) 1994-06-15 CN disclosed
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed